Karam Son

2-(3-Fluoro-4-methylsulfonylaminophenyl)propanamides as Potent Transient Receptor Potential Vanilloid 1 (TRPV1) Antagonists: Structure–Activity Relationships of 2-Amino Derivatives in the<i>N</i>-(6-Trifluoromethylpyridin-3-ylmethyl) C-Region

Myeong Seop Kim, HyungChul Ryu, Dong Wook Kang et al. · Journal of Medicinal Chemistry · 2012 · 41 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +17

2-(3-Fluoro-4-methylsulfonylaminophenyl)propanamides as potent TRPV1 antagonists: Structure activity relationships of the 2-oxy pyridine C-region

Shivaji A. Thorat, Dong Wook Kang, HyungChul Ryu et al. · European Journal of Medicinal Chemistry · 2013 · 22 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +11

TRPV1 antagonist with high analgesic efficacy: 2-Thio pyridine C-region analogues of 2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides

Taehwan Ha, HyungChul Ryu, Sung‐Eun Kim et al. · Bioorganic & Medicinal Chemistry · 2013 · 22 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +14

2-Aryl substituted pyridine C-region analogues of 2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides as highly potent TRPV1 antagonists

HyungChul Ryu, Sejin Seo, Myeong Seop Kim et al. · Bioorganic & Medicinal Chemistry Letters · 2014 · 16 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +6

2-Alkyl/alkenyl substituted pyridine C-region analogues of 2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides as highly potent TRPV1 antagonists

HyungChul Ryu, Sejin Seo, Seong-Hee Cho et al. · Bioorganic & Medicinal Chemistry Letters · 2014 · 14 citations

Pharmacy, Medicinal Chemistry, Pharmacology +7