Shivaji A. Thorat

Structure–activity relationship of human glutaminyl cyclase inhibitors having an N-(5-methyl-1H-imidazol-1-yl)propyl thiourea template

Phuong‐Thao Tran, Van-Hai Hoang, Shivaji A. Thorat et al. · Bioorganic & Medicinal Chemistry · 2013 · 34 citations · Full text

Structure–activity Relationship, Molecular Pharmacology, Biochemistry +12

Discovery of Nonpungent Transient Receptor Potential Vanilloid 1 (TRPV1) Agonist as Strong Topical Analgesic

Jihyae Ann, Ho Shin Kim, Shivaji A. Thorat et al. · Journal of Medicinal Chemistry · 2019 · 34 citations · Full text

Medicinal Chemistry, Trpv1 Agonists, Pain Medicine +13

2-(3-Fluoro-4-methylsulfonylaminophenyl)propanamides as potent TRPV1 antagonists: Structure activity relationships of the 2-oxy pyridine C-region

Shivaji A. Thorat, Dong Wook Kang, HyungChul Ryu et al. · European Journal of Medicinal Chemistry · 2013 · 22 citations · Full text

Biochemistry, Medicine, 2-Oxy Pyridine C-region +6

Pyrazole C-region analogues of 2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides as potent TRPV1 antagonists

Sunho Lee, Changhoon Kim, Jihyae Ann et al. · Bioorganic & Medicinal Chemistry Letters · 2017 · 21 citations · Full text

Medicine, Pharmacological Agent, Pharmacotherapy +3

Discovery of Benzopyridone-Based Transient Receptor Potential Vanilloid 1 Agonists and Antagonists and the Structural Elucidation of Their Activity Shift

Shivaji A. Thorat, Yoonji Lee, Aeran Jung et al. · Journal of Medicinal Chemistry · 2021 · 18 citations · Full text