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TRPV1 antagonist with high analgesic efficacy: 2-Thio pyridine C-region analogues of 2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides

Taehwan Ha, HyungChul Ryu, Sung‐Eun Kim, Ho Shin Kim, Jihyae Ann, Phuong‐Thao Tran, Van-Hai Hoang, Karam Son, Minghua Cui, Sun Choi,

Bioorganic & Medicinal Chemistry · 2013 · 22 citations · 14 references

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14

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Michael J. Caterina, Mark Schumacher, Makoto Tominaga et al. · Nature · 1997 · 9.1K citations

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A peripheral mononeuropathy in rat that produces disorders of pain sensation like those seen in man

Gary J. Bennett, Yuanyu Xie · Pain · 1988 · 5.4K citations

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The Cloned Capsaicin Receptor Integrates Multiple Pain-Producing Stimuli

Makoto Tominaga, Michael J. Caterina, Annika B. Malmberg et al. · Neuron · 1998 · 3.1K citations · Full text

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Vanilloid receptors on sensory nerves mediate the vasodilator action of anandamide

Peter M. Zygmunt, Jesper Petersson, David A. Andersson et al. · Nature · 1999 · 2.1K citations

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Direct activation of capsaicin receptors by products of lipoxygenases: Endogenous capsaicin-like substances

Sun Wook Hwang, Hawon Cho, Jiyeon Kwak et al. · Proceedings of the National Academy of Sciences · 2000 · 1K citations

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