Marian Preston

Discovery of Imidazo[1,2-<i>a</i>]pyridine Ethers and Squaramides as Selective and Potent Inhibitors of Mycobacterial Adenosine Triphosphate (ATP) Synthesis

Subramanyam J. Tantry, Shankar D. Markad, Vikas Shinde et al. · Journal of Medicinal Chemistry · 2017 · 126 citations

Pharmacy, Medicinal Chemistry, Pharmacology +17

Identification and Characterization of Dual Inhibitors of the USP25/28 Deubiquitinating Enzyme Subfamily

Jonathan D.J. Wrigley, Gérald Gavory, Iain Simpson et al. · ACS Chemical Biology · 2017 · 88 citations · Full text

Life Sciences, Biochemistry, Molecular Biology +15

Potent, selective small molecule inhibitors of type III phosphatidylinositol-4-kinase α- but not β-inhibit the phosphatidylinositol signaling cascade and cancer cell proliferation

Michael J. Waring, David Andrews, Paul Faulder et al. · Chemical Communications · 2013 · 34 citations

Life Sciences, Medicinal Chemistry, Pharmacology +15

Generating Selective Leads for Mer Kinase Inhibitors—Example of a Comprehensive Lead-Generation Strategy

J. Willem M. Nissink, Sana Bazzaz, Carolyn Blackett et al. · Journal of Medicinal Chemistry · 2021 · 28 citations · Full text

Pharmacy, Medicinal Chemistry, Oncology +16

A Novel High-Throughput Cell-Based Assay Aimed at Identifying Inhibitors of DNA Metabolism in Bacteria

Jun Fan, Boudewijn L. M. de Jonge, Kathy MacCormack et al. · Antimicrobial Agents and Chemotherapy · 2014 · 22 citations · Full text

Life Sciences, Biotechnology, Molecular Biology +17