Jerzy R. Szewczyk

Discovery of 5-[[4-[(2,3-Dimethyl-2<i>H</i>-indazol-6-yl)methylamino]-2-pyrimidinyl]amino]-2-methyl-benzenesulfonamide (Pazopanib), a Novel and Potent Vascular Endothelial Growth Factor Receptor Inhibitor

Philip A. Harris, Amogh Boloor, Mui Cheung et al. · Journal of Medicinal Chemistry · 2008 · 342 citations · Full text

<i>N</i>-(2-Benzoylphenyl)-<scp>l</scp>-tyrosine PPARγ Agonists. 1. Discovery of a Novel Series of Potent Antihyperglycemic and Antihyperlipidemic Agents

Brad R. Henke, Steven G. Blanchard, Marcus F. Brackeen et al. · Journal of Medicinal Chemistry · 1998 · 299 citations · Full text

Pharmaceutical Science, Pharmacotherapy, Heterocycle Chemistry +17

Regulation of TNF-α secretion by a specific melanocortin-1 receptor peptide agonist

Diane M. Ignar, John L. Andrews, Marilyn Jansen et al. · Peptides · 2003 · 27 citations

Inflammation, Molecular Pharmacology, Signal Transduction +10

An investigation of the absolute configuration of the potent histamine H3 receptor antagonist GT‐2331 using vibrational circular dichroism

Douglas J. Minick, Royston C. B. Copley, Jerzy R. Szewczyk et al. · Chirality · 2007 · 20 citations

Vibrational Circular Dichroism, Chemical Biology, Pharmaceutical Chemistry +20

Discovery of small molecule agonists for the bombesin receptor subtype 3 (BRS-3) based on an omeprazole lead

David L. Carlton, Lissa J. Collin-Smith, Alejandro J. Daniels et al. · Bioorganic & Medicinal Chemistry Letters · 2008 · 18 citations · Full text

Medicinal Chemistry, Drug Target, Biochemistry +12