Ian Hollingsworth

Discovery of a Thiadiazole–Pyridazine-Based Allosteric Glutaminase 1 Inhibitor Series That Demonstrates Oral Bioavailability and Activity in Tumor Xenograft Models

M. Raymond V. Finlay, Mark J. Anderton, Andrew Bailey et al. · Journal of Medicinal Chemistry · 2019 · 29 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +15

Neutral 5-substituted 4-anilinoquinazolines as potent, orally active inhibitors of erbB2 receptor tyrosine kinase

Peter Ballard, Bernard Barlaam, Robert H. Bradbury et al. · Bioorganic & Medicinal Chemistry Letters · 2007 · 25 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +13

Synthesis of Functionalized Cyanopyrazoles via Magnesium Bases

Allan Dishington, J. Lyman Feron, Kathryn Gill et al. · Organic Letters · 2014 · 18 citations

Natural Sciences, Chemistry, Organometallic Chemistry +6

Ring Opening of Cyclic Sulfamidates with Magnesiated Heterocycles: Expedient Synthesis of Highly Functionalised Azaindolines and Azatetrahydroquinolines

Barry R. Hayter, Ian Hollingsworth, Thorsten Nowak · Synlett · 2012 · 18 citations

Natural Sciences, Chemistry, Medicinal Chemistry +16

2-Sulfinyl Oxetanes: Synthesis, Stability and Reactivity

James A. Bull, Kate F. Morgan, Robert Doran et al. · Synlett · 2015 · 16 citations

Pharmacy, Chemistry, Medicinal Chemistry +11