Philip S. Jackson

Multi-step organic synthesis using solid-supported reagents and scavengers: a new paradigm in chemical library generation

Steven V. Ley, Ian R. Baxendale, Robert N. Bream et al. · Journal of the Chemical Society Perkin Transactions 1 · 2000 · 689 citations · Full text

Natural Sciences, Chemical Engineering, Chemistry +13

Discovery of GDC-0077 (Inavolisib), a Highly Selective Inhibitor and Degrader of Mutant PI3Kα

Emily J. Hanan, Marie-Gabrielle Braun, Robert A. Heald et al. · Journal of Medicinal Chemistry · 2022 · 134 citations · Full text

Medicine, Oncology, Pharmacology +14

The Rational Design of Selective Benzoxazepin Inhibitors of the α-Isoform of Phosphoinositide 3-Kinase Culminating in the Identification of ( <i>S</i> )-2-((2-(1-Isopropyl-1 <i>H</i> -1,2,4-triazol-5-yl)-5,6-dihydrobenzo[ <i>f</i> ]imidazo[1,2- <i>d</i> ][1,4]oxazepin-9-yl)oxy)propanamide (GDC-0326)

Timothy P. Heffron, Robert A. Heald, Chudi Ndubaku et al. · Journal of Medicinal Chemistry · 2016 · 106 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +13

Multi‐Step Application of Immobilized Reagents and Scavengers: A Total Synthesis of Epothilone C

Richard Storer, Toshiyasu Takemoto, Philip S. Jackson et al. · Chemistry - A European Journal · 2004 · 85 citations · Full text

Pharmacy, Medicinal Chemistry, Drug Discovery +6

Depressive Disorder in Highly Gifted Adolescents

Philip S. Jackson, Jean Sunde Peterson · Journal of Secondary Gifted Education · 2003 · 84 citations

Social Sciences, Psychiatry, Psychology +17