Xiao‐Shu He

Indoline and piperazine containing derivatives as a novel class of mixed D2/D4 receptor antagonists. Part 2: Asymmetric synthesis and biological evaluation

He Zhao, Xiao‐Shu He, Andrew Thurkauf et al. · Bioorganic & Medicinal Chemistry Letters · 2002 · 56 citations · Full text

Molecular Pharmacology, Derivative (Chemistry), Derivatives +11

Indoline and piperazine containing derivatives as a novel class of mixed D2/D4 receptor antagonists. Part 1: Identification and structure–activity relationships

He Zhao, Andrew Thurkauf, Xiao‐Shu He et al. · Bioorganic & Medicinal Chemistry Letters · 2002 · 24 citations · Full text

Molecular Pharmacology, Derivatives, Biochemistry +10

A new approach to the design of .sigma.-2-selective ligands: synthesis and evaluation of N-[2-(3,4-dichlorophenyl)ethyl]-N-methyl-2-(1-pyrrolidinyl)ethylamine-related polyamines at .sigma.-1 and .sigma.-2 receptor subtypes

Brian R. de Costa, Xiao‐Shu He, Celia Dominguez et al. · Journal of Medicinal Chemistry · 1994 · 19 citations · Full text

Mammalian alkaloids: Synthesis and <i>O</i>‐methylation of (<i>S</i>)‐ and (<i>R</i>)‐3′‐hydroxycoclaurine and their <i>N</i>‐methylated analogues with <i>S</i>‐adenosyl‐<scp>L</scp>‐[<i>methyl</i>‐¹⁴C]methionine in presence of mammalian catechol <i>O</i>‐methyltransferase

Xiao‐Shu He, Dragana Tadić, Małgorzata Brzostowska et al. · Helvetica Chimica Acta · 1991 · 18 citations

Analogs 5A, Bioorganic Chemistry, Mammalian Alkaloids +13

DI-(2,2,2-Trichloroethyl)-Carbonate: Byproduct in Reactions with 2,2,2-Trichloroethyl Chloroformate

Xiao‐Shu He, Arnold Brossi · Synthetic Communications · 1990 · 11 citations

Halogenation, Chemical Engineering, Engineering +8