Gareth M. Davies

AZD9496: An Oral Estrogen Receptor Inhibitor That Blocks the Growth of ER-Positive and <i>ESR1</i> -Mutant Breast Tumors in Preclinical Models

Hazel M. Weir, Robert H. Bradbury, Mandy Lawson et al. · Cancer Research · 2016 · 174 citations

Design and Synthesis of Novel Lactate Dehydrogenase A Inhibitors by Fragment-Based Lead Generation

Richard A. Ward, C. Brassington, Alexander L. Breeze et al. · Journal of Medicinal Chemistry · 2012 · 169 citations · Full text

Aldo-keto Reductase, Molecular Biology, Lead Identification +19

Acoustic Mist Ionization Platform for Direct and Contactless Ultrahigh-Throughput Mass Spectrometry Analysis of Liquid Samples

Ian Sinclair, Martin Bachman, Daniel H. Addison et al. · Analytical Chemistry · 2019 · 117 citations · Full text

Engineering, Analytical Microsystems, Ion Mobility Spectrometry +20

(6S)-6-fluoroshikimic acid, an antibacterial agent acting on the aromatic biosynthetic pathway

Gareth M. Davies, Keith Barrett‐Bee, David A. Jude et al. · Antimicrobial Agents and Chemotherapy · 1994 · 104 citations · Full text

Biosynthesis, Antimicrobial Susceptibility, Biochemistry +15

Methyl-Thiazoles: A Novel Mode of Inhibition with the Potential to Develop Novel Inhibitors Targeting InhA in Mycobacterium tuberculosis

Pravin S. Shirude, Prashanti Madhavapeddi, Maruti Naik et al. · Journal of Medicinal Chemistry · 2013 · 99 citations · Full text

Molecular Biology, Chemical Biology, Enzymatic Modification +19