Brian Bolognese

Monoacidic Inhibitors of the Kelch-like ECH-Associated Protein 1: Nuclear Factor Erythroid 2-Related Factor 2 (KEAP1:NRF2) Protein–Protein Interaction with High Cell Potency Identified by Fragment-Based Discovery

Thomas G. Davies, William E. Wixted, Joseph E. Coyle et al. · Journal of Medicinal Chemistry · 2016 · 306 citations · Full text

Life Sciences, Medicinal Chemistry, Pharmacology +17

Attenuation of Murine Collagen-Induced Arthritis by a Novel, Potent, Selective Small Molecule Inhibitor of IκB Kinase 2, TPCA-1 (2-[(Aminocarbonyl)amino]-5-(4-fluorophenyl)-3-thiophenecarboxamide), Occurs via Reduction of Proinflammatory Cytokines and Antigen-Induced T Cell Proliferation

Patricia L. Podolin, James F. Callahan, Brian Bolognese et al. · Journal of Pharmacology and Experimental Therapeutics · 2004 · 299 citations

Medicine, Immunology, Pharmacology +17

Circadian clock component REV-ERBα controls homeostatic regulation of pulmonary inflammation

Marie Pariollaud, Julie Gibbs, Thomas Hopwood et al. · Journal of Clinical Investigation · 2018 · 205 citations · Full text

Life Sciences, Immunology, Molecular Biology +17

Pharmacological Effects of SB 220025, a Selective Inhibitor of P38 Mitogen-Activated Protein Kinase, in Angiogenesis and Chronic Inflammatory Disease Models

Jeffrey R. Jackson, Brian Bolognese, Leonard M. Hillegass et al. · Journal of Pharmacology and Experimental Therapeutics · 1998 · 174 citations

Medicine, Immunology, Pharmacology +16

A Potent and Selective Nonpeptide Antagonist of CXCR2 Inhibits Acute and Chronic Models of Arthritis in the Rabbit

Patricia L. Podolin, Brian Bolognese, James J. Foley et al. · The Journal of Immunology · 2002 · 162 citations

Medicine, Immunology, Pharmacology +17