Hiromu Habashita

Potent, Low-Molecular-Weight Non-Peptide Inhibitors of Malarial Aspartyl Protease Plasmepsin II

Tasir S. Haque, A. Geoffrey Skillman, Christina E. Lee et al. · Journal of Medicinal Chemistry · 1999 · 168 citations · Full text

A highly stereoselective synthesis of (E)-alkene dipeptide isosteres via organocyanocopper-Lewis acid mediation reaction

Toshiro Ibuka, Hiromu Habashita, Akira Otaka et al. · The Journal of Organic Chemistry · 1991 · 152 citations

Cross-coupling Reaction, Engineering, Alkene Metathesis +13

Novel Low Molecular Weight Spirodiketopiperazine Derivatives Potently Inhibit R5 HIV-1 Infection through Their Antagonistic Effects on CCR5

Kenji Maeda, Kazuhisa Yoshimura, Shiro Shibayama et al. · Journal of Biological Chemistry · 2001 · 126 citations · Full text

A Novel Route to Diastereomerically Pure (<i>E</i>)‐Alkene Dipeptide Isosteres from β‐Aziridinyl‐α,β‐enoates by Treatment with Organocopper Reagents

Toshiro Ibuka, Kazuo Nakai, Hiromu Habashita et al. · Angewandte Chemie International Edition in English · 1994 · 92 citations

Bioorganic Chemistry, Absolute Configuration, Biochemistry +12

Design, Synthesis, and Biological Evaluation of the Combinatorial Library with a New Spirodiketopiperazine Scaffold. Discovery of Novel Potent and Selective Low-Molecular-Weight CCR5 Antagonists

Hiromu Habashita, Masaya Kokubo, Shin-ichi Hamano et al. · Journal of Medicinal Chemistry · 2006 · 79 citations · Full text

Combinatorial Chemistry, Drug Target, Pharmacotherapy +18