Gordafaried Deyanat‐Yazdi

Structure−Activity Relationship Studies of Salinosporamide A (NPI-0052), a Novel Marine Derived Proteasome Inhibitor

Venkat R. Macherla, Scott S. Mitchell, Rama Rao Manam et al. · Journal of Medicinal Chemistry · 2005 · 235 citations

Proteasome Inhibition, Medicinal Chemistry, Pharmaceutical Chemistry +14

Synthesis and Structure–Activity Relationship Study of Antimicrotubule Agents Phenylahistin Derivatives with a Didehydropiperazine-2,5-dione Structure

Yuri Yamazaki, Koji Tanaka, Benjamin Nicholson et al. · Journal of Medicinal Chemistry · 2011 · 104 citations · Full text

Pharmaceutical Science, Organic Chemistry, Microtubule Depolymerization +16

Salinosporamides D−J from the Marine Actinomycete <i>Salinispora tropica</i>, Bromosalinosporamide, and Thioester Derivatives Are Potent Inhibitors of the 20S Proteasome

Katherine A. Reed, Rama Rao Manam, Scott S. Mitchell et al. · Journal of Natural Products · 2007 · 87 citations

Salinosporamides F, Medicinal Chemistry, Marine Biotechnology +15

The Discovery of a Dual TTK Protein Kinase/CDC2-Like Kinase (CLK2) Inhibitor for the Treatment of Triple Negative Breast Cancer Initiated from a Phenotypic Screen

Jennifer R. Riggs, Mark A. Nagy, Jan Elsner et al. · Journal of Medicinal Chemistry · 2017 · 59 citations · Full text

Breast Oncology, Pharmaceutical Chemistry, Tumor Biology +18

Synthetic Lethal Strategy Identifies a Potent and Selective TTK and CLK1/2 Inhibitor for Treatment of Triple-Negative Breast Cancer with a Compromised G1–S Checkpoint

Dan Zhu, Shuichan Xu, Gordafaried Deyanat‐Yazdi et al. · Molecular Cancer Therapeutics · 2018 · 35 citations