In vivo quantification of regional dopamine‐D3 receptor binding potential of (+)‐PHNO: Studies in non‐human primates and transgenic mice

Eugenii A. Rabiner, Mark Slifstein, José N. Nóbrega, +9

Synapse

1,2,4-Triazol-3-yl-thiopropyl-tetrahydrobenzazepines:  A Series of Potent and Selective Dopamine D₃Receptor Antagonists

Fabrizio Micheli, Giorgio Bonanomi, Frank E. Blaney, +37

Journal of Medicinal Chemistry

5-Aryl-4-carboxamide-1,3-oxazoles: Potent and selective GSK-3 inhibitors

Gabriella Gentile, Giancarlo Merlo, Alfonso Pozzan, +11

Bioorganic & Medicinal Chemistry Letters

Medicinal ChemistryMedicineMechanism Of ActionPharmacological AgentPharmacotherapy +4

1,2,4-Triazolyl Azabicyclo[3.1.0]hexanes: A New Series of Potent and Selective Dopamine D₃Receptor Antagonists

Fabrizio Micheli, Luca Arista, Giorgio Bonanomi, +20

Journal of Medicinal Chemistry

Pyrrolo[1,2-a]pyrazine and pyrazolo[1,5-a]pyrazine: Novel, potent, and selective series of Vasopressin1b receptor antagonists

Roberto Arban, Federica Bianchi, Alberto Buson, +9

Bioorganic & Medicinal Chemistry Letters

MedicineMechanism Of ActionPharmacological AgentVasopressin1b Receptor AntagonistsPharmacotherapy +3

Synthesis and Pharmacological Characterization of Novel Druglike Corticotropin-Releasing Factor 1 Antagonists

Romano Di Fabio, Yves St‐Denis, Fabio Maria Sabbatini, +25

Journal of Medicinal Chemistry

Pharmacological CharacterizationNew CrfReceptor AntagonistsPharmacotherapyMolecular Pharmacology +14

Identification and evaluation of [¹¹C]GSK931145 as a novel ligand for imaging the type 1 glycine transporter with positron emission tomography

Jan Passchier, Gabriella Gentile, Rod A. Porter, +6

Synapse

Exploration of the Amine Terminus in a Novel Series of 1,2,4-Triazolo-3-yl-azabicyclo[3.1.0]hexanes as Selective Dopamine D₃Receptor Antagonists

Fabrizio Micheli, Luca Arista, Barbara Bertani, +14

Journal of Medicinal Chemistry

New fused benzazepine as selective D3 receptor antagonists. Synthesis and biological evaluation. Part one: [h]-fused tricyclic systems

Fabrizio Micheli, Giorgio Bonanomi, Simone Braggio, +14

Bioorganic & Medicinal Chemistry Letters

Molecular PharmacologyMedicinal ChemistryPharmaceutical ChemistryHeterocyclicMedicine +9

Identification of 2-(4-pyridyl)thienopyridinones as GSK-3β inhibitors

Gabriella Gentile, Giovanni Bernasconi, Alfonso Pozzan, +10

Bioorganic & Medicinal Chemistry Letters

Molecular PharmacologyMedicinal ChemistryBiochemistryMedicineGsk-3β Inhibitors +6