Concepedia

Takafumi Takai

TT

Statistics

Publications

14

Citations

387

H-Index

13

Active since

2004

Affiliations

Takeda (Japan)(Current)

Takeda (United States)

Takafumi Takai is an author at Takeda (Japan) specializing in drug discovery, medicinal chemistry, and pharmacy.

ORCID

Publications per year

2004–2021

14

Publications

14

Synthesis of a Novel Series of Tricyclic Dihydrofuran Derivatives: Discovery of 8,9-Dihydrofuro[3,2-<i>c</i>]pyrazolo[1,5-<i>a</i>]pyridines as Melatonin Receptor (MT<sub>1</sub>/MT<sub>2</sub>) Ligands

Tatsuki Koike, Takafumi Takai, Yasutaka Hoashi et al. · Journal of Medicinal Chemistry · 2011 · 64 citations · Full text

, , +17

1,6-Dihydro-2<i>H</i>-indeno[5,4-<i>b</i>]furan Derivatives: Design, Synthesis, and Pharmacological Characterization of a Novel Class of Highly Potent MT<sub>2</sub>-Selective Agonists

Tatsuki Koike, Yasutaka Hoashi, Takafumi Takai et al. · Journal of Medicinal Chemistry · 2011 · 49 citations · Full text

, , +16

Discovery of a novel B-cell lymphoma 6 (BCL6)–corepressor interaction inhibitor by utilizing structure-based drug design

Takeshi Yasui, Takeshi Yamamoto, Nozomu Sakai et al. · Bioorganic & Medicinal Chemistry · 2017 · 38 citations · Full text

, , +14

Discovery of 1,2,3,4-tetrahydropyrimido[1,2-a]benzimidazoles as novel class of corticotropin releasing factor 1 receptor antagonists

Takuto Kojima, Michiyo Mochizuki, Takafumi Takai et al. · Bioorganic & Medicinal Chemistry · 2018 · 35 citations · Full text

, , +6

Discovery of a Novel Series of<i>N</i>-Phenylindoline-5-sulfonamide Derivatives as Potent, Selective, and Orally Bioavailable Acyl CoA:Monoacylglycerol Acyltransferase-2 Inhibitors

Kenjiro Sato, Hiroki Takahagi, Takeshi Yoshikawa et al. · Journal of Medicinal Chemistry · 2015 · 30 citations · Full text

, , +14

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