Magda Asselin

Identification, Characterization and Initial Hit-to-Lead Optimization of a Series of 4-Arylamino-3-Pyridinecarbonitrile as Protein Kinase C theta (PKCθ) Inhibitors

Derek C. Cole, Magda Asselin, Agnes Brennan et al. · Journal of Medicinal Chemistry · 2008 · 45 citations · Full text

Tcr Signal Transduction, Drug Target, Inflammatory Lung Disease +19

Inhibition of the Signal Transducer and Activator of Transcription-3 (STAT3) Signaling Pathway by 4-Oxo-1-Phenyl-1,4-Dihydroquinoline-3-Carboxylic Acid Esters

Jun Xu, Derek C. Cole, Chao-Pei Betty Chang et al. · Journal of Medicinal Chemistry · 2008 · 41 citations · Full text

7-Cyano Analogue 8, Chemoprevention Strategy, Cell Death +21

Synthesis and PKCθ inhibitory activity of a series of 4-(indol-5-ylamino)thieno[2,3-b]pyridine-5-carbonitriles

Diane H. Boschelli, Biqi Wu, Ana Carolina Barrios Sosa et al. · Bioorganic & Medicinal Chemistry Letters · 2008 · 33 citations · Full text

Organic Chemistry, Chemistry, Pharmacology +3

The Synthesis and Biological Evaluation of Quinolyl-piperazinyl Piperidines as Potent Serotonin 5-HT_1AAntagonists

Wayne E. Childers, Lisa M. Havran, Magda Asselin et al. · Journal of Medicinal Chemistry · 2010 · 15 citations · Full text

Quinolyl-piperazinyl Piperidines, Molecular Pharmacology, Medicinal Chemistry +13