Jamie D. Knight

[2.2]Paracyclophane derivatives in asymmetric catalysis

Susan E. Gibson, Jamie D. Knight · Organic & Biomolecular Chemistry · 2003 · 287 citations

Architectural Design, Engineering, Heterocyclic +10

Discovery of GDC-0077 (Inavolisib), a Highly Selective Inhibitor and Degrader of Mutant PI3Kα

Emily J. Hanan, Marie-Gabrielle Braun, Robert A. Heald et al. · Journal of Medicinal Chemistry · 2022 · 119 citations · Full text

Oxaziridine-Mediated Amination of Primary Amines:  Scope and Application to a One-Pot Pyrazole Synthesis

Alan Armstrong, Lyn H. Jones, Jamie D. Knight et al. · Organic Letters · 2005 · 96 citations

Noncovalent Mutant Selective Epidermal Growth Factor Receptor Inhibitors: A Lead Optimization Case Study

Robert A. Heald, Krista K. Bowman, Marian C. Bryan et al. · Journal of Medicinal Chemistry · 2015 · 55 citations · Full text

Discovery of a Noncovalent, Mutant-Selective Epidermal Growth Factor Receptor Inhibitor

Bryan Chan, Emily J. Hanan, Krista K. Bowman et al. · Journal of Medicinal Chemistry · 2016 · 32 citations · Full text