Dan Gillie

The discovery of potent blockers of the canonical transient receptor channels, TRPC3 and TRPC6, based on an anilino-thiazole pharmacophore

David G. Washburn, Dennis A. Holt, Jason W. Dodson et al. · Bioorganic & Medicinal Chemistry Letters · 2013 · 58 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +16

Substituted N-{3-[(1,1-dioxido-1,2-benzothiazol-3-yl)(phenyl)amino]propyl}benzamide analogs as potent Kv1.3 ion channel blockers. Part 2

Curt D. Haffner, Stephen A. Thomson, Yu Guo et al. · Bioorganic & Medicinal Chemistry Letters · 2010 · 13 citations · Full text

Natural Sciences, Medicinal Chemistry, Pharmacology +11

N-{3-[(1,1-dioxido-1,2-benzothiazol-3-yl)(phenyl)amino]propyl}benzamide analogs as potent Kv1.3 inhibitors. Part 1

Curt D. Haffner, Stephen A. Thomson, Yu Guo et al. · Bioorganic & Medicinal Chemistry Letters · 2010 · 12 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +6