Matjaž Brvar

Structure-Based Discovery of Substituted 4,5′-Bithiazoles as Novel DNA Gyrase Inhibitors

Matjaž Brvar, Andrej Perdih, M. Renko et al. · Journal of Medicinal Chemistry · 2012 · 177 citations

Crystal Structure, Gyrase B, Molecular Biology +17

Discovery of 4,5,6,7-Tetrahydrobenzo[1,2-<i>d</i>]thiazoles as Novel DNA Gyrase Inhibitors Targeting the ATP-Binding Site

Tihomir Tomašič, Sotirios Katsamakas, Žiga Hodnik et al. · Journal of Medicinal Chemistry · 2015 · 108 citations · Full text

Drug Target, Antibacterial Activity, Bacterial Dna Gyrase +16

Receptor structure-based discovery of non-metabolite agonists for the succinate receptor GPR91

Mette Trauelsen, Elisabeth Rexen Ulven, Siv A. Hjorth et al. · Molecular Metabolism · 2017 · 60 citations · Full text

In silico discovery of 2-amino-4-(2,4-dihydroxyphenyl)thiazoles as novel inhibitors of DNA gyrase B

Matjaž Brvar, Andrej Perdih, Marko Oblak et al. · Bioorganic & Medicinal Chemistry Letters · 2009 · 59 citations

Combinatorial Chemistry, Medicinal Chemistry, Silico Discovery +10

Discovery of substituted oxadiazoles as a novel scaffold for DNA gyrase inhibitors

Žiga Jakopin, Janez Ilaš, Michaela Barančoková et al. · European Journal of Medicinal Chemistry · 2017 · 59 citations · Full text

Combinatorial Chemistry, Medicinal Chemistry, Biochemistry +10