Janez Ilaš

Recent advances in the synthesis of 2H-1,4-benzoxazin-3-(4H)-ones and 3,4-dihydro-2H-1,4-benzoxazines

Janez Ilaš, Marija Sollner Dolenc, D. Kikelj · Tetrahedron · 2005 · 174 citations

Recent Advances, Organic Chemistry, Chemistry +2

Discovery of Benzothiazole Scaffold-Based DNA Gyrase B Inhibitors

Marina Gjorgjieva, Tihomir Tomašič, Michaela Barančoková et al. · Journal of Medicinal Chemistry · 2016 · 140 citations · Full text

Crystal Structure, Medicinal Chemistry, Biochemistry +13

A road map for prioritizing warheads for cysteine targeting covalent inhibitors

Péter Ábrányi‐Balogh, László Petri, Péter A. Szijj et al. · European Journal of Medicinal Chemistry · 2018 · 121 citations

Molecular Docking, Medicinal Chemistry, Covalent Inhibitors +10

Discovery of 4,5,6,7-Tetrahydrobenzo[1,2-<i>d</i>]thiazoles as Novel DNA Gyrase Inhibitors Targeting the ATP-Binding Site

Tihomir Tomašič, Sotirios Katsamakas, Žiga Hodnik et al. · Journal of Medicinal Chemistry · 2015 · 108 citations · Full text

Drug Target, Antibacterial Activity, Bacterial Dna Gyrase +16

3,4-Dihydro-2<i>H</i>-1,4-benzoxazine Derivatives Combining Thrombin Inhibitory and Glycoprotein IIb/IIIa Receptor Antagonistic Activity as a Novel Class of Antithrombotic Compounds with Dual Function

Janez Ilaš, Žiga Jakopin, Tina Borštnar et al. · Journal of Medicinal Chemistry · 2008 · 63 citations · Full text

Thrombin S2, Thrombin Inhibitors, Pharmacotherapy +19