Concepedia
Statistics
Publications
16
Citations
441
H-Index
14
Active since
1999
Affiliations
Xenon Pharmaceuticals (Canada)(Current)
University of Alberta
Novartis (United States)
Shanghai Zhangjiang Laboratory
NAEJA-RGM Pharmaceuticals (Canada)
Shaoyi Sun is an author at Xenon Pharmaceuticals (Canada) specializing in pharmacology, biochemistry, and medicine.
Top concepts
BiochemistryPharmacologyMedicineDrug DiscoveryNatural SciencesPharmacotherapyOrganic ChemistryMedicinal ChemistryChemistryEngineering
Publications per year
1999–2021
A versatile copper-catalyzed coupling reaction of pyridin-2(1H)-ones with aryl halides
Kevin J. Filipski, Jeffrey T. Kohrt, Agustin Casimiro‐Garcia et al. · Tetrahedron Letters · 2006 · 56 citations
Aryl Halides, Chemical Engineering, Cross-coupling Reaction +7
The discovery of benzenesulfonamide-based potent and selective inhibitors of voltage-gated sodium channel Nav1.7
Shaoyi Sun, Qi Jia, Alla Zenova et al. · Bioorganic & Medicinal Chemistry Letters · 2014 · 36 citations · Full text
Tetracyclic spirooxindole blockers of hNaV1.7: activity in vitro and in CFA-induced inflammatory pain model
Sultan Chowdhury, Shifeng Liu, Jay A. Cadieux et al. · Medicinal Chemistry Research · 2012 · 36 citations
Inflammation, Anti-inflammatory, Health Sciences +11
Discovery of Acyl-sulfonamide Na<sub>v</sub>1.7 Inhibitors GDC-0276 and GDC-0310
Brian S. Safina, Steven J. McKerrall, Shaoyi Sun et al. · Journal of Medicinal Chemistry · 2021 · 35 citations · Full text
Identification of Selective Acyl Sulfonamide–Cycloalkylether Inhibitors of the Voltage-Gated Sodium Channel (Na <sub>V</sub> ) 1.7 with Potent Analgesic Activity
Shaoyi Sun, Qi Jia, Alla Zenova et al. · Journal of Medicinal Chemistry · 2018 · 34 citations · Full text
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