Concepedia
Statistics
Publications
18
Citations
695
H-Index
16
Active since
2000
Affiliations
Pfizer (United States)(Current)
Scripps Research Institute
Université Bourgogne Franche-Comté
University of Pittsburgh
Scripps (United States)
Indrawan McAlpine is an author at Pfizer (United States) specializing in organic chemistry, chemistry, and medicine.
Top concepts
MedicineChemistryBiochemistryPharmacologyOrganic ChemistryCatalysisEngineeringDrug DiscoveryNatural SciencesMedicinal Chemistry
Publications per year
2000–2024
Palladium( <scp>ii</scp> )-catalyzed γ-selective hydroarylation of alkenyl carbonyl compounds with arylboronic acids
Rei Matsuura, Tanner C. Jankins, David E. Hill et al. · Chemical Science · 2018 · 78 citations · Full text
Design and Synthesis of Pyridone-Containing 3,4-Dihydroisoquinoline-1(2 <i>H</i> )-ones as a Novel Class of Enhancer of Zeste Homolog 2 (EZH2) Inhibitors
Pei‐Pei Kung, Eugene Rui, Simon Bergqvist et al. · Journal of Medicinal Chemistry · 2016 · 66 citations · Full text
Anti-selective [3+2] (Hetero)annulation of non-conjugated alkenes via directed nucleopalladation
Hui‐Qi Ni, Ilia Kevlishvili, Pranali G. Bedekar et al. · Nature Communications · 2020 · 61 citations · Full text
Discovery of Pyrroloaminopyrazoles as Novel PAK Inhibitors
Chuangxing Guo, Indrawan McAlpine, Junhu Zhang et al. · Journal of Medicinal Chemistry · 2012 · 59 citations · Full text
Medicinal Chemistry, Pharmaceutical Chemistry, Biochemistry +15
Discovery of Allosteric, Potent, Subtype Selective, and Peripherally Restricted TrkA Kinase Inhibitors
Sharan K. Bagal, Kiyoyuki Omoto, David C. Blakemore et al. · Journal of Medicinal Chemistry · 2018 · 52 citations · Full text
Drug Target, Immunology, Molecular Pain +17
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