Fabien Roussel

GDC-9545 (Giredestrant): A Potent and Orally Bioavailable Selective Estrogen Receptor Antagonist and Degrader with an Exceptional Preclinical Profile for ER+ Breast Cancer

Jun Liang, Robert A. Blake, Jae H. Chang et al. · Journal of Medicinal Chemistry · 2021 · 135 citations · Full text

Medicine, Oncology, Pharmacology +15

<i>O</i>-Glycosyl Trichloroacetimidates Bearing Fmoc as Temporary Hydroxy Protecting Group:  A New Access to Solid-Phase Oligosaccharide Synthesis

Fabien Roussel, Laurent Knerr, Matthias Grathwohl et al. · Organic Letters · 2000 · 77 citations

Life Sciences, Biochemistry, Carbohydrate Biochemistry +16

Solid-Phase Synthesis of a Branched Hexasaccharide Using a Highly Efficient Synthetic Strategy

Fabien Roussel, Mohamed Takhi, Richard R. Schmidt · The Journal of Organic Chemistry · 2001 · 66 citations

Life Sciences, Biochemistry, Carbohydrate Biochemistry +16

Identification and optimisation of a series of substituted 5-pyridin-2-yl-thiophene-2-hydroxamic acids as potent histone deacetylase (HDAC) inhibitors

Steve Price, Walter Bordogna, Ruth Braganza et al. · Bioorganic & Medicinal Chemistry Letters · 2006 · 33 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +12

Solid-Phase Synthesis of Lactose-Containing Oligosaccharides

Fabien Roussel, Laurent Knerr, Richard R. Schmidt · European Journal of Organic Chemistry · 2001 · 33 citations

Life Sciences, Biochemistry, Carbohydrate Chemistry +15