Kenneth M. Engstrom

Validation of Diacyl Glycerolacyltransferase I as a Novel Target for the Treatment of Obesity and Dyslipidemia Using a Potent and Selective Small Molecule Inhibitor

Gang Zhao, Andrew J. Souers, Martin J. Voorbach et al. · Journal of Medicinal Chemistry · 2008 · 140 citations · Full text

Life Sciences, Medicinal Chemistry, Pharmacology +17

Implications of the Conformationally Flexible, Macrocyclic Structure of the First-Generation, Direct-Acting Anti-Viral Paritaprevir on Its Solid Form Complexity and Chameleonic Behavior

Ahmad Y. Sheikh, Alessandra Mattei, Rajni M. Bhardwaj et al. · Journal of the American Chemical Society · 2021 · 55 citations

Pharmacy, Medicinal Chemistry, Pharmacology +17

Discovery of adamantane ethers as inhibitors of 11β-HSD-1: Synthesis and biological evaluation

Jyoti Patel, Shuai Qi, Jürgen Dinges et al. · Bioorganic & Medicinal Chemistry Letters · 2006 · 41 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +9

Aminopiperidine indazoles as orally efficacious melanin concentrating hormone receptor-1 antagonists

Anil Vasudevan, Andrew J. Souers, Jennifer C. Freeman et al. · Bioorganic & Medicinal Chemistry Letters · 2005 · 34 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +8

The Stability of <i><i>N</i>,<i>N</i></i>-Carbonyldiimidazole Toward Atmospheric Moisture

Kenneth M. Engstrom, Ahmad Y. Sheikh, Raimundo Ho et al. · Organic Process Research & Development · 2014 · 27 citations

Natural Sciences, Biochemistry, Atmospheric Chemistry +6