Heather M. Madsen

Discovery of PH-797804, a highly selective and potent inhibitor of p38 MAP kinase

Shaun R. Selness, Rajesh Devraj, Balekudru Devadas et al. · Bioorganic & Medicinal Chemistry Letters · 2011 · 72 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +11

Discovery of N-substituted pyridinones as potent and selective inhibitors of p38 kinase

Shaun R. Selness, Rajesh Devraj, Joseph B. Monahan et al. · Bioorganic & Medicinal Chemistry Letters · 2009 · 27 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +12

Discovery of novel spirocyclic inhibitors of fatty acid amide hydrolase (FAAH). Part 1: Identification of 7-azaspiro[3.5]nonane and 1-oxa-8-azaspiro[4.5]decane as lead scaffolds

Marvin J. Meyers, Scott A. Long, Matthew J. Pelc et al. · Bioorganic & Medicinal Chemistry Letters · 2011 · 22 citations

Pharmacy, Medicinal Chemistry, Pharmacology +16

Substituted N-aryl-6-pyrimidinones: A new class of potent, selective, and orally active p38 MAP kinase inhibitors

Balekudru Devadas, Shaun R. Selness, Heather M. Madsen et al. · Bioorganic & Medicinal Chemistry Letters · 2011 · 22 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +9

Prevalent Polymorphisms in Wild-Type HIV-1 Integrase Are Unlikely To Engender Drug Resistance to Dolutegravir (S/GSK1349572)

Cindy Vavro, Samiul Hasan, Heather M. Madsen et al. · Antimicrobial Agents and Chemotherapy · 2013 · 19 citations · Full text

Life Sciences, Molecular Biology, Molecular Genetics +17