Gabriella Traquandi

3-Aminopyrazole Inhibitors of CDK2/Cyclin A as Antitumor Agents. 1. Lead Finding

Paolo Pevarello, Maria Gabriella Brasca, Raffaella Amici et al. · Journal of Medicinal Chemistry · 2004 · 157 citations · Full text

Drug Target, Lead Identification, Pharmacotherapy +23

Identification of <i>N</i>,1,4,4-Tetramethyl-8-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4,5-dihydro-1<i>H</i>-pyrazolo[4,3-<i>h</i>]quinazoline-3-carboxamide (PHA-848125), a Potent, Orally Available Cyclin Dependent Kinase Inhibitor

Maria Gabriella Brasca, Nadia Amboldi, Dario Ballinari et al. · Journal of Medicinal Chemistry · 2009 · 125 citations · Full text

Drug Target, Chemoprevention Strategy, Gynecology +18

3-Aminopyrazole Inhibitors of CDK2/Cyclin A as Antitumor Agents. 2. Lead Optimization

Paolo Pevarello, Maria Gabriella Brasca, Paolo Orsini et al. · Journal of Medicinal Chemistry · 2005 · 107 citations · Full text

Chemoprevention Strategy, Pharmacotherapy, Chemical Biology +20

Identification of Potent Pyrazolo[4,3-<i>h</i>]quinazoline-3-carboxamides as Multi-Cyclin-Dependent Kinase Inhibitors

Gabriella Traquandi, Marina Ciomei, Dario Ballinari et al. · Journal of Medicinal Chemistry · 2010 · 40 citations · Full text

Compound 59, Molecular Pharmacology, Medicinal Chemistry +14

Synthesis and preliminary biological evaluation of new α-amino amide anticonvulsants incorporating a dextromethorphan moiety

Paolo Pevarello, Gabriella Traquandi, A. Bonsignori et al. · Bioorganic & Medicinal Chemistry Letters · 1999 · 10 citations · Full text

Dextromethorphan Moiety, Pharmaceutical Science, Preliminary Biological Evaluation +7