Neil Westlund

Barriers to rotation about the chiral axis of tertiary aromatic amides

Anjum Ahmed, Ryan A. Bragg, Jonathan Clayden et al. · Tetrahedron · 1998 · 188 citations

Chiral Axis, Engineering, Tertiary Aromatic Amides +6

Discovery of 3-(3-(4-(1-Aminocyclobutyl)phenyl)-5-phenyl-3<i>H</i>-imidazo[4,5-<i>b</i>]pyridin-2-yl)pyridin-2-amine (ARQ 092): An Orally Bioavailable, Selective, and Potent Allosteric AKT Inhibitor

Jean‐Marc Lapierre, Sudharshan Eathiraj, David Vensel et al. · Journal of Medicinal Chemistry · 2016 · 105 citations · Full text

Pharmaceutical Science, Pharmacotherapy, Pharmaceutical Chemistry +18

Discovery and Optimization of a Series of 3-(3-Phenyl-3<i>H</i>-imidazo[4,5-<i>b</i>]pyridin-2-yl)pyridin-2-amines: Orally Bioavailable, Selective, and Potent ATP-Independent Akt Inhibitors

Mark A. Ashwell, Jean‐Marc Lapierre, Christopher J. Brassard et al. · Journal of Medicinal Chemistry · 2012 · 98 citations · Full text

Chemical Biology, Pharmaceutical Chemistry, Biophysical Screening Strategy +19

Synthesis of the Kopsia alkaloids (±)-pauciflorine B, (±)-lahadinine B, (±)-kopsidasine, (±)-kopsidasine-N-oxide, (±)-kopsijasminilam and (±)-11-methoxykopsilongine

Philip Magnus, Lewis Gazzard, L. Hobson et al. · Tetrahedron · 2002 · 88 citations

-Pauciflorine B, Bioorganic Chemistry, -Lahadinine B +7

Atroposelectivity in the reactions of ortholithiated aromatic tertiary amides with aldehydes

Peter Bowles, Jonathan Clayden, Madeleine Helliwell et al. · Journal of the Chemical Society Perkin Transactions 1 · 1997 · 73 citations

Cross-coupling Reaction, Novel Organocatalysts, Engineering +12