Bharat Lagu

Identification of NVP-TNKS656: The Use of Structure–Efficiency Relationships To Generate a Highly Potent, Selective, and Orally Active Tankyrase Inhibitor

Michael D. Shultz, Atwood K. Cheung, C.A. Kirby et al. · Journal of Medicinal Chemistry · 2013 · 122 citations · Full text

Drug Target, Selective Tankyrase Inhibitors, Pharmacotherapy +18

Novel highly selective inhibitors of ubiquitin specific protease 30 (USP30) accelerate mitophagy

Arthur F. Kluge, Bharat Lagu, Pranab Maiti et al. · Bioorganic & Medicinal Chemistry Letters · 2018 · 122 citations · Full text

Protease Inhibitors, Cell Autophagy, Mitophagy +8

Design and Synthesis of Novel α₁_a Adrenoceptor-Selective Antagonists. 1. Structure−Activity Relationship in Dihydropyrimidinones

Dhanapalan Nagarathnam, Shou Wu Miao, Bharat Lagu et al. · Journal of Medicinal Chemistry · 1999 · 112 citations · Full text

Organic Chemistry, Pharmacotherapy, Chemistry +16

Discovery of NVP‐LEQ506, a Second‐Generation Inhibitor of Smoothened

Stefan Peukert, Feng He, Miao Dai et al. · ChemMedChem · 2013 · 88 citations

Molecular Pharmacology, Continued Optimization, Competitor Compound +15

Stereo- and regioselective synthesis of chiral diamines and triamines from pseudoephedrine and ephedrine

R. Karl Dieter, Niranjan Deo, Bharat Lagu et al. · The Journal of Organic Chemistry · 1992 · 66 citations

Altmetric Attention Score, Karl Dieter, Organic Chemistry +9