Geoffrey W. Mellor

High Throughput Fluorescence Polarization: A Homogeneous Alternative to Radioligand Binding for Cell Surface Receptors

Michael Allen, J.J. Reeves, Geoffrey W. Mellor · SLAS DISCOVERY · 2000 · 101 citations · Full text

5-(1H-Benzimidazol-1-yl)-3-alkoxy-2-thiophenecarbonitriles as potent, selective, inhibitors of IKK-ε kinase

Paul Bamborough, J.A. Christopher, Geoffrey J. Cutler et al. · Bioorganic & Medicinal Chemistry Letters · 2006 · 51 citations · Full text

Molecular Pharmacology, Medicinal Chemistry, Ikk-ε Kinase +5

Rational design of 4-amino-5,6-diaryl-furo[2,3-d]pyrimidines as potent glycogen synthase kinase-3 inhibitors

Yasushi Miyazaki, Yutaka Maeda, Hideyuki Sato et al. · Bioorganic & Medicinal Chemistry Letters · 2008 · 50 citations · Full text

Combinatorial Chemistry, Medicinal Chemistry, Biochemistry +8

A polyclonal antibody preparation with Michaelian catalytic properties

Gerard Gallacher, Caroline S. Jackson, Mark Searcey et al. · Biochemical Journal · 1991 · 44 citations · Full text

Ionization characteristics of the Cys-25/His-159 interactive system and of the modulatory group of papain: resolution of ambiguity by electronic perturbation of the quasi-2-mercaptopyridine leaving group in a new pyrimidyl disulphide reactivity probe

Geoffrey W. Mellor, Emrys W. Thomas, Christopher M. Topham et al. · Biochemical Journal · 1993 · 37 citations · Full text

Engineering, Pka Value, Biochemistry +12