Susan M. Westaway

8-Substituted Pyrido[3,4-<i>d</i>]pyrimidin-4(3<i>H</i>)-one Derivatives As Potent, Cell Permeable, KDM4 (JMJD2) and KDM5 (JARID1) Histone Lysine Demethylase Inhibitors

Vassilios Bavetsias, Rachel M. Lanigan, G.F. Ruda et al. · Journal of Medicinal Chemistry · 2016 · 98 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +16

GSK962040: a small molecule, selective motilin receptor agonist, effective as a stimulant of human and rabbit gastrointestinal motility

Gareth J. Sanger, Susan M. Westaway, Ashley Barnes et al. · Neurogastroenterology & Motility · 2009 · 77 citations

Medicine, Medicinal Chemistry, Pharmacology +16

Cell Penetrant Inhibitors of the KDM4 and KDM5 Families of Histone Lysine Demethylases. 2. Pyrido[3,4-<i>d</i>]pyrimidin-4(3<i>H</i>)-one Derivatives

Susan M. Westaway, Alex Preston, Michael D. Barker et al. · Journal of Medicinal Chemistry · 2016 · 67 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +9

Cell Penetrant Inhibitors of the KDM4 and KDM5 Families of Histone Lysine Demethylases. 1. 3-Amino-4-pyridine Carboxylate Derivatives

Susan M. Westaway, Alex Preston, Michael D. Barker et al. · Journal of Medicinal Chemistry · 2016 · 59 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +15

Assessing histone demethylase inhibitors in cells: lessons learned

Stephanie B. Hatch, Clarence Yapp, Raquel Carvalho Montenegro et al. · Epigenetics & Chromatin · 2017 · 52 citations · Full text

Life Sciences, Molecular Biology, Pharmacology +13