Albert Gyorkos

The total synthesis of (.+-.)-epi-jatrophone and (.+-.)-jatrophone using palladium-catalyzed carbonylative coupling of vinyl triflates with vinyl stannanes as the macrocycle-forming step

Albert Gyorkos, J. K. Stille, Louis S. Hegedus · Journal of the American Chemical Society · 1990 · 116 citations

Materials Science, Chemical Engineering, Cross-coupling Reaction +15

Development of Orally Active Nonpeptidic Inhibitors of Human Neutrophil Elastase

Kazuyuki Ohmoto, Tetsuya Yamamoto, Motohiro Okuma et al. · Journal of Medicinal Chemistry · 2001 · 64 citations · Full text

Pharmaceutical Science, Bioorganic Chemistry, Immunology +17

Design and Synthesis of New Orally Active Nonpeptidic Inhibitors of Human Neutrophil Elastase

Kazuyuki Ohmoto, Tetsuya Yamamoto, Toshihide Horiuchi et al. · Journal of Medicinal Chemistry · 2000 · 56 citations · Full text

Molecular Pharmacology, Medicinal Chemistry, Antimicrobial Drug Discovery +15

Design and Synthesis of Benzimidazoles As Novel Corticotropin-Releasing Factor 1 Receptor Antagonists

Michiyo Mochizuki, Masakuni Kori, Katsumi Kobayashi et al. · Journal of Medicinal Chemistry · 2016 · 18 citations · Full text

Combinatorial Chemistry, Pharmaceutical Science, Receptor Antagonists +17

Biochemical Characterization of α-Ketooxadiazole Inhibitors of Elastases

Maciej Wieczorek, Albert Gyorkos, Lyle W. Spruce et al. · Archives of Biochemistry and Biophysics · 1999 · 12 citations

Biochemistry, Medicine, α-Ketooxadiazole Inhibitors +5