Vishal Unadkat

Synthesis and structure–activity relationship of potent, selective and orally active anthranilamide-based factor Xa inhibitors: Application of weakly basic sulfoximine group as novel S4 binding element

Vrajesh B. Pandya, Mukul R. Jain, Ganes Chakrabarti et al. · European Journal of Medicinal Chemistry · 2012 · 41 citations · Full text

Structure–activity Relationship, Medicinal Chemistry, Biochemistry +10

Design, Synthesis of Novel, Potent, Selective, Orally Bioavailable Adenosine A_2AReceptor Antagonists and Their Biological Evaluation

Sujay Basu, Dinesh A. Barawkar, Sachin Thorat et al. · Journal of Medicinal Chemistry · 2017 · 22 citations · Full text

Bioisosteric replacement of dihydropyrazole of 4S-(−)-3-(4-chlorophenyl)-N-methyl-N′-[(4-chlorophenyl)-sulfonyl]-4-phenyl-4,5-dihydro-1H-pyrazole-1-caboxamidine (SLV-319) a potent CB1 receptor antagonist by imidazole and oxazole

Brijesh Kumar Srivastava, Rina Soni, Amit Joharapurkar et al. · Bioorganic & Medicinal Chemistry Letters · 2007 · 13 citations

Bioisosteric Replacement, Molecular Pharmacology, Bioorganic Chemistry +10

Rational design-aided discovery of novel 1,2,4-oxadiazole derivatives as potential EGFR inhibitors

Vishal Unadkat, Shishir Rohit, Paranjay Parikh et al. · Bioorganic Chemistry · 2021 · 12 citations

Combinatorial Chemistry, Medicinal Chemistry, Biochemistry +10