Ester Colarusso

Targeting mPGES-1 by a Combinatorial Approach: Identification of the Aminobenzothiazole Scaffold to Suppress PGE₂ Levels

Maria Giovanna Chini, Assunta Giordano, Marianna Potenza et al. · ACS Medicinal Chemistry Letters · 2020 · 25 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +13

Identification of 2,4,5-trisubstituted-2,4-dihydro-3H-1,2,4-triazol-3-one-based small molecules as selective BRD9 binders

Ester Colarusso, Sara Ceccacci, Maria Chiara Monti et al. · European Journal of Medicinal Chemistry · 2022 · 15 citations · Full text

Pharmacy, Chemistry, Medicinal Chemistry +9

Exploring the chemical space of functionalized [1,2,4]triazolo[4,3-a]quinoxaline-based compounds targeting the bromodomain of BRD9

Erica Gazzillo, Martina Pierri, Ester Colarusso et al. · Bioorganic Chemistry · 2023 · 13 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +17

Essential Oils of Laurus nobilis L.: From Chemical Analysis to In Silico Investigation of Anti-Inflammatory Activity by Soluble Epoxide Hydrolase (sEH) Inhibition

Francesca Fantasma, Vadym Samukha, Michela Aliberti et al. · Foods · 2024 · 11 citations · Full text

Life Sciences, Biochemistry, Botany +15

Thiazolidin-4-one-based compounds interfere with the eicosanoid biosynthesis pathways by mPGES-1/sEH/5-LO multi-target inhibition

Ester Colarusso, Marianna Potenza, Gianluigi Lauro et al. · European Journal of Medicinal Chemistry Reports · 2022 · 10 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +17