Erica Gazzillo

Introducing structure-based three-dimensional pharmacophore models for accelerating the discovery of selective BRD9 binders

Martina Pierri, Erica Gazzillo, Maria Giovanna Chini et al. · Bioorganic Chemistry · 2021 · 16 citations

Pharmacy, Medicinal Chemistry, Pharmacology +14

Identification of 2,4,5-trisubstituted-2,4-dihydro-3H-1,2,4-triazol-3-one-based small molecules as selective BRD9 binders

Ester Colarusso, Sara Ceccacci, Maria Chiara Monti et al. · European Journal of Medicinal Chemistry · 2022 · 15 citations · Full text

Pharmacy, Chemistry, Medicinal Chemistry +9

Exploring the chemical space of functionalized [1,2,4]triazolo[4,3-a]quinoxaline-based compounds targeting the bromodomain of BRD9

Erica Gazzillo, Martina Pierri, Ester Colarusso et al. · Bioorganic Chemistry · 2023 · 13 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +17

Repositioning of Quinazolinedione-Based Compounds on Soluble Epoxide Hydrolase (sEH) through 3D Structure-Based Pharmacophore Model-Driven Investigation

Erica Gazzillo, Stefania Terracciano, Dafne Ruggiero et al. · Molecules · 2022 · 10 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +14

6‐Methylquinazolin‐4(3<i>H</i>)‐one Based Compounds as BRD9 Epigenetic Reader Binders: A Rational Combination of <i>in silico</i> Studies and Chemical Synthesis

Ester Colarusso, Erica Gazzillo, Eleonora Boccia et al. · European Journal of Organic Chemistry · 2022 · 10 citations

Pharmacy, Medicinal Chemistry, Pharmacology +17