John J. McAtee

Design and Optimization of Sulfone Pyrrolidine Sulfonamide Antagonists of Transient Receptor Potential Vanilloid-4 with in Vivo Activity in a Pulmonary Edema Model

Joseph E. Pero, Jay M. Matthews, David J. Behm et al. · Journal of Medicinal Chemistry · 2018 · 34 citations · Full text

Palosuran inhibits binding to primate UT receptors in cell membranes but demonstrates differential activity in intact cells and vascular tissues

David J. Behm, John J. McAtee, Jason W. Dodson et al. · British Journal of Pharmacology · 2008 · 31 citations · Full text

Discovery of GSK3527497: A Candidate for the Inhibition of Transient Receptor Potential Vanilloid-4 (TRPV4)

Carl Brooks, Linda S. Barton, David J. Behm et al. · Journal of Medicinal Chemistry · 2019 · 23 citations · Full text

Identification, Synthesis, and Characterization of a Major Circulating Human Metabolite of TRPV4 Antagonist GSK2798745

Joseph E. Pero, John J. McAtee, David J. Behm et al. · ACS Medicinal Chemistry Letters · 2021 · 20 citations · Full text

Aminomethylpiperazines as selective urotensin antagonists

Mark A. Hilfiker, Daohua Zhang, Sarah E. Dowdell et al. · Bioorganic & Medicinal Chemistry Letters · 2008 · 13 citations · Full text

Selective Urotensin Antagonists, Urology, Medicine +6