Jacek Malinowski

Isolation and studies of the mutagenic activity in the Ames test of flavonoids naturally occurring in medical herbs

Hanna Czeczot, Barbara Tudek, J. Kusztelak et al. · Mutation Research/Genetic Toxicology · 1990 · 165 citations

Polyphenolics, Medical Herbs, Mutagenic Activity +8

Unusual 4-hydroxybenzaldehyde synthase activity from tissue cultures of the vanilla orchid Vanilla planifolia

Andrzej Podstolski, Daphna Havkin‐Frenkel, Jacek Malinowski et al. · Phytochemistry · 2002 · 95 citations

Biosynthesis, Engineering, Biochemistry +6

Inhibitors of Human Immunodeficiency Virus Type 1 (HIV-1) Attachment. 12. Structure–Activity Relationships Associated with 4-Fluoro-6-azaindole Derivatives Leading to the Identification of 1-(4-Benzoylpiperazin-1-yl)-2-(4-fluoro-7-[1,2,3]triazol-1-yl-1<i>H</i>-pyrrolo[2,3-<i>c</i>]pyridin-3-yl)ethane-1,2-dione (BMS-585248)

Alicia Regueiro‐Ren, Qiufen Xue, Jacob J. Swidorski et al. · Journal of Medicinal Chemistry · 2013 · 50 citations

Vitro Potency, Good Potency, Azaindole Core +17

A new catalytic activity from tobacco converting 2‐coumaric acid to salicylic aldehyde

Jacek Malinowski, Magdalena Krzymowska, K. Godon et al. · Physiologia Plantarum · 2007 · 22 citations

Phytoalexin, New Catalytic Activity, Biosynthesis +12

Utilization of in vitro Caco‐2 permeability and liver microsomal half‐life screens in discovering BMS‐488043, a novel HIV‐1 attachment inhibitor with improved pharmacokinetic properties

Zheng Yang, Lisa Zadjura, Anthony M. Marino et al. · Journal of Pharmaceutical Sciences · 2009 · 22 citations

Improved Pharmacokinetic Properties, Vitro Caco‐2 Permeability, Medicine +9