Mohamed H. El‐Shershaby

From triazolophthalazines to triazoloquinazolines: A bioisosterism-guided approach toward the identification of novel PCAF inhibitors with potential anticancer activity

Mohamed H. El‐Shershaby, Adel Ghiaty, Ashraf H. Bayoumi et al. · Bioorganic & Medicinal Chemistry · 2021 · 67 citations · Full text

Medicinal Chemistry, Biochemistry, Novel Pcaf Inhibitors +11

The antimicrobial potential and pharmacokinetic profiles of novel quinoline-based scaffolds: synthesis and <i>in silico</i> mechanistic studies as dual DNA gyrase and DHFR inhibitors

Mohamed H. El‐Shershaby, Kamal M. El‐Gamal, Ashraf H. Bayoumi et al. · New Journal of Chemistry · 2021 · 64 citations

Pathogenic Microbes, Available Antimicrobial Agents, Dhfr Inhibitors +22

1,2,4-Triazolo[4,3-<i>c</i>]quinazolines: a bioisosterism-guided approach towards the development of novel PCAF inhibitors with potential anticancer activity

Mohamed H. El‐Shershaby, Adel Ghiaty, Ashraf H. Bayoumi et al. · New Journal of Chemistry · 2021 · 46 citations

Novel Pcaf Inhibitors, Potential Anticancer Activity, Pharmacotherapy +25

Synthesis, antimicrobial evaluation, DNA gyrase inhibition, and in silico pharmacokinetic studies of novel quinoline derivatives

Mohamed H. El‐Shershaby, Kamal M. El‐Gamal, Ashraf H. Bayoumi et al. · Archiv der Pharmazie · 2020 · 44 citations