Publication | Closed Access
1,2,4-Triazolo[4,3-<i>c</i>]quinazolines: a bioisosterism-guided approach towards the development of novel PCAF inhibitors with potential anticancer activity
46
Citations
37
References
2021
Year
Novel Pcaf InhibitorsPotential Anticancer ActivityPharmacotherapyPharmaceutical ChemistryTumor BiologyMolecular PharmacologyMedicinal ChemistrySmall Inhibitor MoleculesAnti-cancer AgentRadiation OncologyCancer ResearchMedicineBioisosterism-guided ApproachTumor TargetingTargeted TherapyDrug DevelopmentPotential Therapeutic StrategyPharmacologyCancer TreatmentTumor MicroenvironmentBiomolecular EngineeringDrug TargetingNatural SciencesRational Drug DesignImmune Checkpoint InhibitorOncologySmall MoleculesDrug Discovery
Targeting PCAF with small inhibitor molecules has emerged as a potential therapeutic strategy for the treatment of cancer.
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