Concepedia

Jan Heeres

JH

Statistics

Publications

39

Citations

3.1K

H-Index

23

Active since

1969

Affiliations

Janssen (Belgium)(Current)

University of Antwerp

Johnson & Johnson (United States)

Instituut voor Tropische Geneeskunde

Rutgers, The State University of New Jersey

Jan Heeres is an author at Janssen (Belgium) specializing in pharmacology, medicinal chemistry, and drug discovery.

Publications per year

1969–2017

39

Publications

39

Roles of Conformational and Positional Adaptability in Structure-Based Design of TMC125-R165335 (Etravirine) and Related Non-nucleoside Reverse Transcriptase Inhibitors That Are Highly Potent and Effective against Wild-Type and Drug-Resistant HIV-1 Variants

Kalyan Das, Arthur D. Clark, Paul Lewi et al. · Journal of Medicinal Chemistry · 2004 · 511 citations

, , +17

Antimycotic imidazoles. Part 4. Synthesis and antifungal activity of ketoconazole, a new potent orally active broad-spectrum antifungal agent

Jan Heeres, L. J. J. Backx, J. H. Mostmans et al. · Journal of Medicinal Chemistry · 1979 · 341 citations

, , +14

TMC125, a Novel Next-Generation Nonnucleoside Reverse Transcriptase Inhibitor Active against Nonnucleoside Reverse Transcriptase Inhibitor-Resistant Human Immunodeficiency Virus Type 1

Koen Andries, Hilde Azijn, Theo Thielemans et al. · Antimicrobial Agents and Chemotherapy · 2004 · 322 citations · Full text

, , +17

Preparation and antimycotic properties of derivatives of 1-phenethylimidazole

Erik F. Godefroi, Jan Heeres, J. Van Cutsem et al. · Journal of Medicinal Chemistry · 1969 · 266 citations

, , +6

SYNOPSIS:  SYNthesize and OPtimize System in Silico

H. Maarten Vinkers, Marc R. de Jonge, Frederik F. D. Daeyaert et al. · Journal of Medicinal Chemistry · 2003 · 229 citations · Full text

, , +15

1–5 of 39