Scott H. Watterson

Discovery of 6-Fluoro-5-(<i>R</i>)-(3-(<i>S</i>)-(8-fluoro-1-methyl-2,4-dioxo-1,2-dihydroquinazolin-3(4<i>H</i>)-yl)-2-methylphenyl)-2-(<i>S</i>)-(2-hydroxypropan-2-yl)-2,3,4,9-tetrahydro-1<i>H</i>-carbazole-8-carboxamide (BMS-986142): A Reversible Inhibitor of Bruton’s Tyrosine Kinase (BTK) Conformationally Constrained by Two Locked Atropisomers

Scott H. Watterson, George V. De Lucca, Qing Shi et al. · Journal of Medicinal Chemistry · 2016 · 142 citations · Full text

The Total Synthesis of (±)-Ginkgolide B

Michael T. Crimmins, Jennifer M. Pace, Philippe G. Nantermet et al. · Journal of the American Chemical Society · 2000 · 105 citations

Medicinal Chemistry, Ginkgolide B, Bioorganic Chemistry +13

Discovery of Branebrutinib (BMS-986195): A Strategy for Identifying a Highly Potent and Selective Covalent Inhibitor Providing Rapid in Vivo Inactivation of Bruton’s Tyrosine Kinase (BTK)

Scott H. Watterson, Qingjie Liu, Myra Beaudoin Bertrand et al. · Journal of Medicinal Chemistry · 2019 · 104 citations · Full text

Tyrosine Kinase, Immunology, Quantitative Pharmacology +20

(Phenylsulfonyl)allenes as Substrates for Cycloaddition Reactions: Intramolecular Cyclizations onto Unactivated Alkenes

Albert Padwa, Michael Meske, S. Shaun Murphree et al. · Journal of the American Chemical Society · 1995 · 75 citations

Intramolecular Cyclizations, Molecular Sciences, Engineering +9

Phenylsulfonyl Ene−Allenes as Efficient Precursors to Bicyclic Systems via Intramolecular [2 + 2]-Cycloaddition Reactions

Albert Padwa, Helmut Lipka, Scott H. Watterson et al. · The Journal of Organic Chemistry · 2003 · 65 citations