Concepedia
Statistics
Publications
5
Citations
641
H-Index
Active since
2000
Affiliations
Station Biologique de Roscoff(Current)
National Cancer Institute
Universität Hamburg
Centre National de la Recherche Scientifique
Technische Universität Braunschweig
Maryse Leost is an author at Station Biologique de Roscoff specializing in pharmacology, drug discovery, and medicine.
Top concepts
PharmacologyMedicineBiochemistryDrug DiscoveryCell SignalingChemical BiologyDrug DevelopmentNatural SciencesMolecular DockingMedicinal Chemistry
Publications per year
2000–2005
Paullones are potent inhibitors of glycogen synthase kinase‐3β and cyclin‐dependent kinase 5/p25
Maryse Leost, Christiane Schultz, Andreas Link et al. · European Journal of Biochemistry · 2000 · 370 citations · Full text
Independent actions on cyclin-dependent kinases and aryl hydrocarbon receptor mediate the antiproliferative effects of indirubins
Marie Knockaert, Marc Blondel, Stéphane Bach et al. · Oncogene · 2004 · 97 citations
Signal Transduction, Cyclin-dependent Kinases, Biochemistry +10
Evaluation and Comparison of 3D-QSAR CoMSIA Models for CDK1, CDK5, and GSK-3 Inhibition by Paullones
Conrad Kunick, Kathrin Lauenroth, Karen Wieking et al. · Journal of Medicinal Chemistry · 2003 · 97 citations · Full text
Epoxide-containing side chains enhance antiproliferative activity of paullones
Xu Xie, Thomas Lemcke, Rick Gussio et al. · European Journal of Medicinal Chemistry · 2005 · 39 citations
Pharmacology, Epoxide-containing Side Chains, Antimicrobial Compound
Structure‐Aided Optimization of Kinase Inhibitors Derived from Alsterpaullone
Conrad Kunick, Zhihong Zeng, Rick Gussio et al. · ChemBioChem · 2005 · 38 citations · Full text
Molecular Docking, Molecular Pharmacology, Medicinal Chemistry +15
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