Abdulsalam A. M. Alkhaldi

3-Methylthiazolo[3,2-a]benzimidazole-benzenesulfonamide conjugates as novel carbonic anhydrase inhibitors endowed with anticancer activity: Design, synthesis, biological and molecular modeling studies

Abdulsalam A. M. Alkhaldi, Mohammad M. Al‐Sanea, Alessio Nocentini et al. · European Journal of Medicinal Chemistry · 2020 · 78 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +16

Functional analysis of drug resistance‐associated mutations in the <scp><i>T</i></scp><i>rypanosoma brucei</i> adenosine transporter 1 (<scp>TbAT</scp>1) and the proposal of a structural model for the protein

Jane C. Munday, Daniel N. A. Tagoe, Anthonius A. Eze et al. · Molecular Microbiology · 2015 · 57 citations · Full text

Medicine, Genetics, Molecular Genetics +15

Synthesis and Structure–Activity Analysis of New Phosphonium Salts with Potent Activity against African Trypanosomes

Andrea Taladriz‐Sender, Alan R. Healy, Eddysson J. Flores Pérez et al. · Journal of Medicinal Chemistry · 2012 · 56 citations

Pharmacy, Medicinal Chemistry, Pharmacology +17

Symmetrical choline-derived dications display strong anti-kinetoplastid activity

Hasan M. S. Ibrahim, Mohammed I. Al-Salabi, Nasser El Sabbagh et al. · Journal of Antimicrobial Chemotherapy · 2010 · 46 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +17

Trypanocidal action of bisphosphonium salts through a mitochondrial target in bloodstream form Trypanosoma brucei

Abdulsalam A. M. Alkhaldi, Jan Martínek, Brian Panicucci et al. · International Journal for Parasitology Drugs and Drug Resistance · 2015 · 46 citations · Full text

Life Sciences, Biochemistry, Pharmacology +16