Satoki Doi

Broad Antiretroviral Activity and Resistance Profile of the Novel Human Immunodeficiency Virus Integrase Inhibitor Elvitegravir (JTK-303/GS-9137)

Kazuya Shimura, Eiichi Kodama, Yasuko Sakagami et al. · Journal of Virology · 2007 · 343 citations · Full text

Medicine, Human Retrovirus, Immunology +15

Discovery of Conformationally Constrained Tetracyclic Compounds as Potent Hepatitis C Virus NS5B RNA Polymerase Inhibitors

Kazutaka Ikegashira, Takahiro Oka, Shintaro Hirashima et al. · Journal of Medicinal Chemistry · 2006 · 110 citations · Full text

Combinatorial Chemistry, Biochemistry, Medicine +11

SAR Exploration Guided by LE and Fsp ³ : Discovery of a Selective and Orally Efficacious RORγ Inhibitor

Kazuyuki Hirata, Masayuki Kotoku, Noriyoshi Seki et al. · ACS Medicinal Chemistry Letters · 2015 · 58 citations · Full text

Discovery of a Janus Kinase Inhibitor Bearing a Highly Three-Dimensional Spiro Scaffold: JTE-052 (Delgocitinib) as a New Dermatological Agent to Treat Inflammatory Skin Disorders

Satoru Noji, Yoshinori Hara, Tomoya Miura et al. · Journal of Medicinal Chemistry · 2020 · 52 citations · Full text

Discovery of Second Generation RORγ Inhibitors Composed of an Azole Scaffold

Masayuki Kotoku, Takaki Maeba, Shingo Fujioka et al. · Journal of Medicinal Chemistry · 2019 · 31 citations · Full text

Butanoic Acid Scaffold, Immunology, Chemical Biology +20