Edwin B. Villhauer

1-[[(3-Hydroxy-1-adamantyl)amino]acetyl]-2-cyano-(<i>S</i>)-pyrrolidine:  A Potent, Selective, and Orally Bioavailable Dipeptidyl Peptidase IV Inhibitor with Antihyperglycemic Properties

Edwin B. Villhauer, J. A. Brinkman, Goli B. Naderi et al. · Journal of Medicinal Chemistry · 2003 · 609 citations · Full text

Molecular Pharmacology, Medicinal Chemistry, Pharmaceutical Science +14

NVP-DPP728 (1-[[[2-[(5-Cyanopyridin-2-yl)amino]ethyl]amino]acetyl]-2-cyano-(<i>S</i>)-pyrrolidine), a Slow-Binding Inhibitor of Dipeptidyl Peptidase IV

Thomas E. Hughes, Manisha Mone, Mary E. Russell et al. · Biochemistry · 1999 · 125 citations

Molecular Pharmacology, Medicinal Chemistry, Pharmaceutical Chemistry +14

1-[2-[(5-Cyanopyridin-2-yl)amino]ethylamino]acetyl-2-(<i>S</i>)-pyrrolidinecarbonitrile:  A Potent, Selective, and Orally Bioavailable Dipeptidyl Peptidase IV Inhibitor with Antihyperglycemic Properties

Edwin B. Villhauer, J. A. Brinkman, Goli B. Naderi et al. · Journal of Medicinal Chemistry · 2002 · 120 citations · Full text

Pharmaceutical Science, Peptide Science, Pharmacotherapy +18

Conformation of [1-13C,15N]Acetyl-L-carnitine. Rotational-Echo, Double-Resonance Nuclear Magnetic Resonance Spectroscopy

Robert C. Anderson, Terry Gullion, James M. Joers et al. · Journal of the American Chemical Society · 1995 · 50 citations

Engineering, Biochemistry, Donut Icon +14

A Concise Synthesis of a Novel Insulin-Like Growth Factor I Receptor (IGF-IR) Inhibitor

Joel Slade, Joginder S. Bajwa, Hui Liu et al. · Organic Process Research & Development · 2007 · 38 citations

Concise Synthesis, Medicinal Chemistry, Growth Hormone +13