Francesco Rianjongdee

Design and Synthesis of a Highly Selective and <i>In Vivo</i>-Capable Inhibitor of the Second Bromodomain of the Bromodomain and Extra Terminal Domain Family of Proteins

Alex Preston, Stephen J. Atkinson, Paul Bamborough et al. · Journal of Medicinal Chemistry · 2020 · 53 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +14

Discovery of a Highly Selective BET BD2 Inhibitor from a DNA-Encoded Library Technology Screening Hit

Francesco Rianjongdee, Stephen J. Atkinson, Chun‐wa Chung et al. · Journal of Medicinal Chemistry · 2021 · 45 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +14

Template-Hopping Approach Leads to Potent, Selective, and Highly Soluble Bromo and Extraterminal Domain (BET) Second Bromodomain (BD2) Inhibitors

Helen Aylott, Stephen J. Atkinson, Paul Bamborough et al. · Journal of Medicinal Chemistry · 2021 · 28 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +14

Fragment-based Scaffold Hopping: Identification of Potent, Selective, and Highly Soluble Bromo and Extra Terminal Domain (BET) Second Bromodomain (BD2) Inhibitors

Jonathan T. Seal, Stephen J. Atkinson, Paul Bamborough et al. · Journal of Medicinal Chemistry · 2021 · 24 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +17

Automated LC-MS analysis and data extraction for high-throughput chemistry

J. S. Mason, Harry Wilders, David J. Fallon et al. · Digital Discovery · 2023 · 23 citations · Full text

Natural Sciences, Chemistry, Analytical Chemistry +10