Enzo Tramontano

Classification and characterization of human endogenous retroviruses; mosaic forms are common

Laura Vargiu, Patricia Rodriguez‐Tomé, Göran Sperber et al. · Retrovirology · 2016 · 318 citations · Full text

Geometrically and Conformationally Restrained Cinnamoyl Compounds as Inhibitors of HIV-1 Integrase:  Synthesis, Biological Evaluation, and Molecular Modeling

Marino Artico, Roberto Di Santo, Roberta Costi et al. · Journal of Medicinal Chemistry · 1998 · 162 citations · Full text

Combinatorial Chemistry, Hiv-1 Integrase, Enzyme Assays +17

Identification of Inhibitors of SARS-CoV-2 3CL-Pro Enzymatic Activity Using a Small Molecule in Vitro Repurposing Screen

Maria Kuzikov, Elisa Costanzi, Jeanette Reinshagen et al. · ACS Pharmacology & Translational Science · 2021 · 154 citations · Full text

In vitro selection and molecular characterization of human immunodeficiency virus-1 resistant to non-nucleoside inhibitors of reverse transcriptase.

John W. Mellors, Ginger E. Dutschman, Guang‐Jin Im et al. · Molecular Pharmacology · 1992 · 131 citations

6-[1-(4-Fluorophenyl)methyl-1H-pyrrol-2-yl)]-2,4-dioxo-5-hexenoic acid ethyl ester a novel diketo acid derivative which selectively inhibits the HIV-1 viral replication in cell culture and the ribonuclease H activity in vitro

Enzo Tramontano, Francesca Esposito, Roberta Badas et al. · Antiviral Research · 2005 · 117 citations

Medicinal Chemistry, Viral Replication, Hiv-1 Viral Replication +13