Holia Hatoum‐Mokdad

Discovery of AZD9833, a Potent and Orally Bioavailable Selective Estrogen Receptor Degrader and Antagonist

James S. Scott, Amber Balazs, Bernard Barlaam et al. · Journal of Medicinal Chemistry · 2020 · 111 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +17

Synthesis and structure activity relationships of novel small molecule cathepsin D inhibitors

Jacques Dumas, David R. Brittelli, Jinshan Chen et al. · Bioorganic & Medicinal Chemistry Letters · 1999 · 88 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +12

1-Phenyl-5-pyrazolyl ureas: potent and selective p38 kinase inhibitors

Jacques Dumas, Holia Hatoum‐Mokdad, Robert Sibley et al. · Bioorganic & Medicinal Chemistry Letters · 2000 · 53 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +7

A novel estrogen receptor ligand template

Robert Sibley, Holia Hatoum‐Mokdad, Robert Schoenleber et al. · Bioorganic & Medicinal Chemistry Letters · 2003 · 36 citations · Full text

Life Sciences, Biochemistry, Molecular Biology +11

Discovery of Efficacious <i>Pseudomonas aeruginosa</i>-Targeted Siderophore-Conjugated Monocarbams by Application of a Semi-mechanistic Pharmacokinetic/Pharmacodynamic Model

Kerry E. Murphy-Benenato, Pratik Bhagunde, April Chen et al. · Journal of Medicinal Chemistry · 2015 · 27 citations

Medicine, Medicinal Chemistry, Pharmacology +17