C. Lerner

A Convergent Enantioselective Route to Structurally Diverse 6-Deoxytetracycline Antibiotics

Mark G. Charest, C. Lerner, Jason D. Brubaker et al. · Science · 2005 · 294 citations

Enantioselective Synthesis, Bioorganic Chemistry, Engineering +11

A Robust Platform for the Synthesis of New Tetracycline Antibiotics

Cuixiang Sun, Qiu Wang, Jason D. Brubaker et al. · Journal of the American Chemical Society · 2008 · 128 citations · Full text

A Real-World Perspective on Molecular Design

Bernd Kuhn, Wolfgang Guba, Jérôme Hert et al. · Journal of Medicinal Chemistry · 2016 · 119 citations · Full text

Drug Target, Hit Identification, Molecular Biology +20

Machine learning-powered antibiotics phenotypic drug discovery

Sannah Zoffmann, Maarten Vercruysse, Fethallah Benmansour et al. · Scientific Reports · 2019 · 107 citations · Full text

Safety screening in early drug discovery: An optimized assay panel

Stefanie Bendels, Caterina Bissantz, Bernhard Fasching et al. · Journal of Pharmacological and Toxicological Methods · 2019 · 78 citations

Drug Safety, Predictive Toxicology, Preclinical Drug Evaluation +10