Eliezer Falb

<i>In situ</i> generation of Fmoc‐amino acid chlorides using <i>bis</i>‐(trichloromethyl)carbonate and its utilization for difficult couplings in solid‐phase peptide synthesis

Eliezer Falb, Tamar Yechezkel, Yoseph Salitra · Journal of Peptide Research · 1999 · 145 citations

Difficult Couplings, Bioorganic Chemistry, Engineering +17

Acetyl Chloride-Methanol as a Convenient Reagent for: A) Quantitative Formation of Amine Hydrochlorides B) Carboxylate Ester Formation C) Mild Removal of N-t-Boc-Protective Group.

Ayelet Nudelman, Yosi Bechor, Eliezer Falb et al. · Synthetic Communications · 1998 · 107 citations

Mild Removal, Chemical Engineering, Engineering +15

A highly efficient Suzuki–Miyaura methylation of pyridines leading to the drug pirfenidone and its CD₃ version (SD-560)

Eliezer Falb, Konstantin Ulanenko, Andrey Tor et al. · Green Chemistry · 2017 · 42 citations

Quantitative Suzuki–miyaura Routes, Medicinal Chemistry, Pharmaceutical Chemistry +12

A Convenient Synthesis of Chiral Oxazolidin-2-Ones and Thiazolidin-2-Ones and an Improved Preparation of Triphosgene

Eliezer Falb, Abraham Nudelman · Synthetic Communications · 1993 · 41 citations

Internal Cooling System, Engineering, Free Acids +11

IOOC Route to Substituted Chiral Pyrrolidines. Potential Glycosidase Inhibitors

Eliezer Falb, Yosi Bechor, Abraham Nudelman et al. · The Journal of Organic Chemistry · 1998 · 38 citations

Medicinal Chemistry, Natural Product Synthesis, Amino Acids +12