Publication | Closed Access
A highly efficient Suzuki–Miyaura methylation of pyridines leading to the drug pirfenidone and its CD<sub>3</sub> version (SD-560)
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Citations
37
References
2017
Year
Quantitative Suzuki–miyaura RoutesMedicinal ChemistryPharmaceutical ChemistryDerivative (Chemistry)BiochemistryNatural SciencesMedicineOrganic ChemistryEfficient Suzuki–miyaura MethylationHeterocycle ChemistryPharmacologyDrug PirfenidoneFirst Methylation/deuteromethylationBiomolecular EngineeringDrug Discovery
The first methylation/deuteromethylation in green and nearly quantitative Suzuki–Miyaura routes to pirfenidone and its d<sub>3</sub> analog SD-560, at 99% isotopic purity.
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