Michel Garneau

Structure−Activity Study on a Novel Series of Macrocyclic Inhibitors of the Hepatitis C Virus NS3 Protease Leading to the Discovery of BILN 2061

Montse Llinàs‐Brunet, Murray D. Bailey, Gordon T. Bolger et al. · Journal of Medicinal Chemistry · 2004 · 186 citations

Competitive Hexapeptide Inhibitors, Pharmacotherapy, Antiviral Drug +16

Discovery of BI 224436, a Noncatalytic Site Integrase Inhibitor (NCINI) of HIV-1

Lee D. Fader, Éric Malenfant, Mathieu Parisien et al. · ACS Medicinal Chemistry Letters · 2014 · 175 citations · Full text

Hiv-1 Integrase, Immunology, Molecular Biology +16

A potent peptidomimetic inhibitor of HSV ribonucleotide reductase with antiviral activity in vivo

Michel Liuzzi, Robert Déziel, Nell Moss et al. · Nature · 1994 · 132 citations

Molecular Virology, Antiviral Agents, Antiviral Activity +12

Preclinical Characterization of BI 201335, a C-Terminal Carboxylic Acid Inhibitor of the Hepatitis C Virus NS3-NS4A Protease

Peter W. White, Montse Llinàs‐Brunet, Ma’an Amad et al. · Antimicrobial Agents and Chemotherapy · 2010 · 109 citations · Full text

Immunology, Molecular Biology, Antiviral Drug +16

Preclinical Profile of BI 224436, a Novel HIV-1 Non-Catalytic-Site Integrase Inhibitor

Craig Fenwick, Ma’an Amad, Murray D. Bailey et al. · Antimicrobial Agents and Chemotherapy · 2014 · 98 citations · Full text